Vol 13, No 4(52) (2015)

Full Issue

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Table of Contents

The synthesis of 1,5-diaryl-4-arylthiopyrrolidin-2-ones by arylsulfenylation of styryl acetic acid N-arylamides PDF
N. M. Tsyzoryk, I. Yu. Danyliuk, A. I. Vaskevych, R. I. Vaskevych, M. V. Vovk 3-5
Methylation of position 8 in the pyridine moiety of the N-(benzyl)-2-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide molecule as an attempt to enhance their analgesic properties PDF
I. V. Ukrainets, O. V. Gorokhova, L. V. Sydorenko, S. G. Taran 6-11
A convenient way of 3-fluoro-1,8-naphthalimide synthesis PDF
N. F. Fedko, V. F. Anikin 12-15
Testing of a new docking scoring function on the example of inhibitors of protein tyrosine phosphatase 1B PDF
V. Yu. Tanchuk, V. O. Tanin 16-19
Synthesis and the antimicrobial activity of 3-(2-methyl-4-oxo-1,4-dihydroquinoline-3-yl)propanoic acids PDF
V. O. Zubkov, T. P. Osolodchenko, N. I. Ruschak, O. L. Kamenetska, O. V. Kiz 20-26
The synthesis and anticancer properties of 2-(4-amino-5-methyl-4H-[1,2,4]triazol-3-ylsulfanyl)-N-(5-R-benzylthiazol-2-yl)-acetamides PDF
Yu. V. Ostapiuk, V. S. Matiychuk, M. D. Obushak 27-31
The synthesis, reactivity and the antimicrobial activity of substituted thieno[2,3-d]pyrimidine-4(3H)-thio(seleno)nes PDF
D. O. Kolomieitsev, V. I. Markov, V. O. Astakhina, S. I. Kovalenko, S. A. Varenichenko, O. V. Kharchenko 32-38
The study of regularities of the structure – analgesic activity relationship in a series of 4-hydroxy-Nn-(pyridin-2-yl)-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamides PDF
I. V. Ukrainets, L. A. Petrushova, O. V. Gorokhova, O. O. Davydenko 39-43
The complexing ability of n-substituted thiourea derivatives as chelating ligands in the reaction with PdCl2 PDF
Yu. L. Zborovskii, V. V. Orysyk, D. O. Melnychenko, S. I. Orysyk, H. H. Repich, L. V. Garmanchuk, L. I. Palchykovska, V. I. Pekhnyo, M. V. Vovk 44-49
5,6-Dihydro-[1,2,4]triazolo[1,5-c]quinazolines. Message 1. Features of interactions between [2-(3-aryl-1H-1,2,4-triazole-5-yl)phenyl]amines, aliphatic and aromatic aldehydes PDF
S. V. Kholodnyak, K. P. Schabelnyk, O. Yu. Voskoboynik, G. G. Berest, S. I. Kovalenko 50-56
The synthesis and evaluation of the bactericidal activity of 4-(4-chloro-1H-imidazol-5-yl)-2-oxo-1,2-dihydropyridin-3-carbonitriles PDF (Українська)
O. Ya. Mel’nyk, V. O. Chornous, N. D. Yakovychuk, N. V. Mel’nichenko, M. V. Vovk 57-61
Development and validation of the method for determination of related impurities in riboxin tablets PDF
M. V. Rosada, N. Yu. Bevz, V. A. Georgiyants 62-67
The study of retention regularities for the potential drug substances of 1,2,4-triazol-3-ylthioacetic acids and their salts series by the method of HPLC/DAD-MS PDF (Українська)
B. O. Varynskyi, Ye. G. Knysh, V. V. Parchenko, A. G. Kaplaushenko 68-75